Naltriben mesylate

Tocris Bioscience, part of Bio-Techne | Catalog # 0892

Standard δ2 selective antagonist
Discontinued Product
0892 has been discontinued. View all delta Opioid Receptor Antagonists products.

Key Product Details

Description

Standard δ2 selective antagonist

View all delta Opioid Receptor Antagonists »

Product Description

Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively). Displays selectivity for the δ2 subtype in vivo.

Licensing Information

Sold with the permission of the University of Minnesota

Product Specifications

Molecular Weight

511.59

Formula

C26H25NO4.CH3SO3H

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinan mesylate

CAS Number

122517-78-6

PubChem ID

45073482

InChI Key

XRRFZOCDAWPIBB-IDRHMUJXSA-N

SMILES

C[S](O)(=O)=O.[H][C@@]12OC3=C(O)C=CC4=C3[C@@]11CCN(CC3CC3)[C@]([H])(C4)[C@]1(O)CC1=C2OC2=C1C=CC=C2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 25.58 50 with gentle warming

Preparing Stock Solutions for Naltriben mesylate

The following data is based on the product molecular weight 511.59

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.5 mM 3.91 mL 19.55 mL 39.09 mL
2.5 mM 0.78 mL 3.91 mL 7.82 mL
5 mM 0.39 mL 1.95 mL 3.91 mL
25 mM 0.08 mL 0.39 mL 0.78 mL

Calculators

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for Naltriben mesylate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Naltriben mesylate

For research use only

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