CYM 5520
Tocris Bioscience, part of Bio-Techne | Catalog # 5418
Selective S1P2 allosteric agonist
Key Product Details
Description
Selective S1P2 allosteric agonist
Product Description
CYM 5520 is a selective S1P2 allosteric agonist (EC50 = 0.48 μM). Selective for S1P2 receptors over a panel of 29 other receptors and transporters.Product Specifications
Molecular Weight
345.39
Formula
C21H19N3O2
Storage
Store at +4°C
Purity
≥98% (HPLC)
Chemical Name
1-[2-[2,5-Dimethyl-1-(phenylmethyl)-1H-pyrrol-3-yl]-2-oxoethyl]-1,6-dihydro-6-oxo-3-pyridinecarbonitrile
CAS Number
1449747-00-5
PubChem ID
25110470
InChI Key
FMYGNANMYYHBSU-UHFFFAOYSA-N
SMILES
CC1=C(C(CN3C=C(C#N)C=CC3=O)=O)C=C(C)N1CC2=CC=CC=C2
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 34.54 | 100 |
Preparing Stock Solutions
for CYM 5520
The following data is based on the product molecular weight 345.39
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.90 mL | 14.48 mL | 28.95 mL |
| 5 mM | 0.58 mL | 2.90 mL | 5.79 mL |
| 10 mM | 0.29 mL | 1.45 mL | 2.90 mL |
| 50 mM | 0.06 mL | 0.29 mL | 0.58 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Satsu A sphingosine 1-phosphate receptor 2 selective allosteric agonist. Bioorg.Med.Chem. 2013 PMID: 23849205
Product Specific Notices for CYM 5520
For research use only
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