CYM 50769
Tocris Bioscience, part of Bio-Techne | Catalog # 4948
Novel non-peptide NPBWR1 antagonist
Key Product Details
Description
Novel non-peptide NPBWR1 antagonist
Alternative Names
ML250
Product Description
CYM 50769 is a novel non-peptide antagonist of neuropeptide W/B receptor 1 (NPBWR1, GPR7) (IC50 = 0.12 μM).Product Specifications
Molecular Weight
416.86
Formula
C24H17ClN2O3
Storage
Store at +4°C
Purity
≥98% (HPLC)
Chemical Name
5-Chloro-2-(9H-fluoren-9-yl)-4-(4-methoxyphenoxy)-3(2H)-pyridazinone
CAS Number
1421365-63-0
PubChem ID
50904505
InChI Key
QHVSQUYCVUHYKT-UHFFFAOYSA-N
SMILES
ClC(C=N4)=C(OC5=CC=C(OC)C=C5)C(N4C2C3=C(C=CC=C3)C1=CC=CC=C12)=O
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 41.69 | 100 |
Preparing Stock Solutions
for CYM 50769
The following data is based on the product molecular weight 416.86
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.40 mL | 11.99 mL | 23.99 mL |
| 5 mM | 0.48 mL | 2.40 mL | 4.80 mL |
| 10 mM | 0.24 mL | 1.20 mL | 2.40 mL |
| 50 mM | 0.05 mL | 0.24 mL | 0.48 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Guerrero SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists. Bioorg.Med.Chem.Lett. 2013 PMID: 23287738
Product Specific Notices for CYM 50769
For research use only
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