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CP 339818 hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 1399

Non-peptide, potent KV1.3 channel blocker
Discontinued Product
1399 has been discontinued. View all Voltage-gated Potassium Channel Blockers products.

Key Product Details

Description

Non-peptide, potent KV1.3 channel blocker

Product Description

CP 339818 hydrochloride is a potent, non-peptide KV1.3 channel antagonist that preferentially binds to the C-type inactivated state of the channel (IC50 ~ 200 nM) . Inhibits KV1.4 with an IC50 of ~ 300 nM. Selective over KV1.1, KV1.2, KV1.5, KV1.6, KV3.1-4, and KV4.2.

Product Specifications

Molecular Weight

340.89

Formula

C21H24N2.HCl

Storage

Store at RT

Purity

≥99% (HPLC)

Chemical Name

N-[1-(Phenylmethyl)-4(1H)-quinolinylidene]-1 pentanamine hydrochloride

CAS Number

478341-55-8

PubChem ID

20761468

InChI Key

JIRISCAPZWLWCG-UHFFFAOYSA-N

SMILES

CCCCC\N=C2C1=CC=CC=C1N(CC3=CC=CC=C3)C=C/2.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 20

Preparing Stock Solutions for CP 339818 hydrochloride

The following data is based on the product molecular weight 340.89

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.2 mM 14.67 mL 73.34 mL 146.67 mL
1 mM 2.93 mL 14.67 mL 29.33 mL
2 mM 1.47 mL 7.33 mL 14.67 mL
10 mM 0.29 mL 1.47 mL 2.93 mL

Calculators

Molarity Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for CP 339818 hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CP 339818 hydrochloride

For research use only

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