CGP 52432

Tocris Bioscience, part of Bio-Techne | Catalog # 1246

Potent and selective GABAB antagonist
Catalog #
Availability
Size / Price
Qty
1246/10
1246/50
Print Quote
Bulk Order
100% Guarantee

Key Product Details

Description

Potent and selective GABAB antagonist

View all GABA-B Receptor Antagonists »

Product Description

CGP 52432 is a potent, selective GABAB receptor antagonist (IC50 = 85 nM).

Licensing Information

Sold with the permission of Novartis Pharma AG

Product Specifications

Molecular Weight

384.24

Formula

C15H24Cl2NO4P

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

3-[[(3,4-Dichlorophenyl)methyl]amino]propyl] diethoxymethyl)phosphinic acid

CAS Number

139667-74-6

PubChem ID

132252

InChI Key

GJZVQXWEIYRHBE-UHFFFAOYSA-N

SMILES

ClC1=CC=C(CNCCCP(C(OCC)OCC)(O)=O)C=C1Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 1.92 5

Preparing Stock Solutions for CGP 52432

The following data is based on the product molecular weight 384.24

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.05 mM 52.05 mL 260.25 mL 520.51 mL
0.25 mM 10.41 mL 52.05 mL 104.10 mL
0.5 mM 5.21 mL 26.03 mL 52.05 mL
2.5 mM 1.04 mL 5.21 mL 10.41 mL

Calculators

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Dilution Calculator

Calculate the dilution required to prepare a stock solution.

x
=
x

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Background References

References are publications that support the biological activity of the product.

Product Documents for CGP 52432

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CGP 52432

For research use only

Privacy Policy
Cookie Policy
Site Map
© Copyright 2026 Bio-Techne. All Rights Reserved. All trademarks and registered trademarks are the property of Bio-Techne and its brands unless otherwise specified.