CGP 12177 hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 1134

β3 partial agonist. β1/β2 antagonist
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Key Product Details

Description

β3 partial agonist. β1/β2 antagonist

View all Adrenergic beta-3 Receptor Agonists »

Product Description

CGP 12177 hydrochloride is a partial agonist at β3-adrenoceptors. β1- and β2-adrenoceptor antagonist (Ki values are 0.9, 4 and 88 nM for β1, β2 and β3 receptors respectively).

Product Specifications

Molecular Weight

315.80

Formula

C14H21N3O3.HCl

Storage

Store at RT

Chemical Name

4-[3-[(1,1-Dimethylethyl)amino]2-hydroxypropoxy]-1,3-dihydro-2H-benzimidazol-2-one hydrochloride

CAS Number

64208-32-8

PubChem ID

11957517

InChI Key

YQVFCYCTITZLSX-UHFFFAOYSA-N

SMILES

Cl.CC(C)(C)NCC(O)COC1=CC=CC2=C1NC(=O)N2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 50

Preparing Stock Solutions for CGP 12177 hydrochloride

The following data is based on the product molecular weight 315.80

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.5 mM 6.33 mL 31.67 mL 63.33 mL
2.5 mM 1.27 mL 6.33 mL 12.67 mL
5 mM 0.63 mL 3.17 mL 6.33 mL
25 mM 0.13 mL 0.63 mL 1.27 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for CGP 12177 hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CGP 12177 hydrochloride

For research use only

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