Bay 59-3074

Tocris Bioscience, part of Bio-Techne | Catalog # 2500

CB1/CB2 receptor partial agonist
Discontinued Product
2500 has been discontinued. View all Non-selective Cannabinoid Receptor Agonists products.

Key Product Details

Description

CB1/CB2 receptor partial agonist

View all Non-selective Cannabinoid Receptor Agonists »

Product Description

Bay 59-3074 is a novel CB1/CB2 receptor partial agonist (Ki values are 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively). Orally active CB1 agonist in vivo. Displays anti-hyperalgesic and antiallodynic properties in rat models of chronic neuropathic and inflammatory pain.

Licensing Information

Sold for research purposes under agreement from Bayer

Product Specifications

Molecular Weight

453.35

Formula

C18H13F6NO4S

Storage

Store at +4°C

Purity

≥99% (HPLC)

Chemical Name

3-[2-Cyano-3-(trifluoromethyl)phenoxy]phenyl 4,4,4-trifluoro-1-butanesulfonic acid ester

CAS Number

406205-74-1

PubChem ID

10479060

InChI Key

LWUSZIVDPJPVBW-UHFFFAOYSA-N

SMILES

FC(F)(F)CCCS(=O)(=O)OC1=CC(OC2=CC=CC(=C2C#N)C(F)(F)F)=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 45.34 100
Ethanol 45.34 100

Preparing Stock Solutions for Bay 59-3074

The following data is based on the product molecular weight 453.35

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.21 mL 11.03 mL 22.06 mL
5 mM 0.44 mL 2.21 mL 4.41 mL
10 mM 0.22 mL 1.10 mL 2.21 mL
50 mM 0.04 mL 0.22 mL 0.44 mL

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Product Documents for Bay 59-3074

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Bay 59-3074

For research use only

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